Patent · US Expired

4-substituted anthracyclinones and their preparation

US5218130A · kind A · utility

5Cited by
6References
7Claims
0Family size

Assignee

Inventors

Key dates

Filing dateJan 25, 1991
Grant dateJun 8, 1993
Priority date
Expiry dateJan 25, 2011

Classification

  • Technology area (CPC A)Human Necessities
  • CPC primaryA61P31/04
  • WIPO fieldOrganic fine chemistry
  • WIPO sectorChemistry

Abstract

4-substituted anthracyclinones of formula (I) ##STR1## wherein R represents a hydrogen atom or a straight or branched alkyl, alkenyl or alkynyl group having from 1 to 10 carbon atoms, are intermediates in the preparation of antitumor anthracycline glycosides of formula (IX): ##STR2## wherein R is as defined above and R.sub.1 is a hydrogen atom or a hydroxy group, and pharmaceutically acceptable salts thereof.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.