Patent · US Expired

Azacyclic carboxylic acid derivatives and their preparation and use

US5229404A · kind A · utility

0Cited by
5References
20Claims
0Family size

Assignee

Inventors

Key dates

Filing dateDec 6, 1991
Grant dateJul 20, 1993
Priority date
Expiry dateDec 6, 2011

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07D409/14
  • WIPO fieldOrganic fine chemistry
  • WIPO sectorChemistry

Abstract

Novel O-alkylated oximes of the general formula I ##STR1## wherein R.sup.1 and R.sup.2 are optionally substituted aromatic or heteroaromatic rings, R.sup.3 is hydrogen or lower alkyl, R.sup.4 is a nitrogen containing, substituted ring or an amino group carrying a substituted ring, and n and m independently are 0, 1 or 2, are potent inhibitors of GABA re-uptake from the synaptic cleft.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.