Patent · US Expired

2-aza-2-desamino analogues of 5,8-dideazafolic acid

US5234925A · kind A · utility

0Cited by
6References
11Claims
0Family size

Assignee

Inventor

Key dates

Filing dateAug 14, 1991
Grant dateAug 10, 1993
Priority date
Expiry dateAug 14, 2011

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07D417/12
  • WIPO fieldOrganic fine chemistry
  • WIPO sectorChemistry

Abstract

2-Aza-2-desamino analogues of 5,8-dideazafolic acid, which analogues have the formula ##STR1## wherein X is an aryl or heteroaryl moiety; PA1 R.sup.1 is H, C.sub.1 -C.sub.4 alkyl, C.sub.3 -C.sub.4 alkenyl, or C.sub.3 -C.sub.4 alkynyl; and PA1 R.sup.2 is OH, an L-.alpha.-amino acid, or a peptide comprising L-.alpha.-amino acids.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.