Patent · US Expired

Inhibitors of platelet-derived growth factor

US5238950A · kind A · utility

89Cited by
3References
12Claims
0Family size

Assignee

Inventors

Key dates

Filing dateDec 17, 1991
Grant dateAug 24, 1993
Priority date
Expiry dateDec 17, 2011

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07D487/04
  • WIPO fieldOrganic fine chemistry
  • WIPO sectorChemistry

Abstract

A method of inhibiting the binding of PDGF using compounds of the formula I ##STR1## useful in the treatment of atherosclerosis, cancer, retinal detachment, pulmonary fibrosis, arthritis, psoriasis and glomerulonephritis, and restenosis following angioplasty or vascular surgery is disclosed. Also disclosed are pharmaceutical compositions and novel PDGF inhibitory compounds of the formula ##STR2## or a pharmaceutically acceptable addition salt thereof, useful in the treatment of atherosclerosis, cancer, retinal detachment, pulmonary fibrosis, arthritis, psoriasis and glomerulonephritis, and restenosis following angioplasty or vascular surgery.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.