Patent · US Expired

Carbonate intermediates for the synthesis of purine substituted cyclopentene derivatives

US5241069A · kind A · utility

2Cited by
3References
2Claims
0Family size

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Key dates

Filing dateNov 6, 1991
Grant dateAug 31, 1993
Priority date
Expiry dateNov 6, 2011

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07D473/18
  • WIPO fieldOrganic fine chemistry
  • WIPO sectorChemistry

Abstract

This invention relates to the new process for preparing the 1R-cis isomer of carbovir, (1R-cis)-amino-1,9-dihydro-9-[4-(hydroxymethyl)-2-cyclopenten-1-yl]-6H-pur in-6-one, an antiviral agent and intermediates of the formula (Vlb) use in that process ##STR1## wherein X is chloro, bromo or iodo and R is (C.sub.1-6) alkyl.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.