Patent · US Expired

Heterocyclic compounds which have useful pharmaceutical utility

US5264436A · kind A · utility

0Cited by
2References
16Claims
0Family size

Assignee

Inventors

Key dates

Filing dateSep 16, 1991
Grant dateNov 23, 1993
Priority date
Expiry dateSep 16, 2011

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07D403/06
  • WIPO fieldOrganic fine chemistry
  • WIPO sectorChemistry

Abstract

A compound of formula (I): ##STR1## or a pharmaceutically acceptable salt, ester or amide thereof, or a pharmaceutically acceptable solvate thereof, wherein: PA1 Z represents a residue of a substituted or unsubstituted aryl group, PA1 A.sub.1 represents a substituted or unsubstituted methylene group or a substituted or unsubstituted ethylene group; PA1 A.sub.2 represents a substituted or unsubstituted methylene group or a substituted or unsubstituted ethylene group; PA1 providing that at least one of A.sup.1 or A.sup.2 represents a substituted methylene group or a substituted ethylene group, PA1 X represents O or NR.sup.o wherein R.sup.o represents a hydrogen atom, a substituted or unsubstituted alkyl group, a substituted or unsubstituted aryl group, an alkanoyl group substituted or unsubstituted in the alkyl moiety, or an arylalkyl moiety substituted or unsubstituted in the aryl moiety, PA1 p represents an integer 2 or 3, and PA1 q represents an integer in the range of from 1 to 12; a process for preparing such a compound, a composition comprising such a compound and the use of such a compound in medicine.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.