Patent · US Expired

0-hydroxyethyl and acyloxyethyl derivatives of [ser].sup.8 cyclosporins

US5284826A · kind A · utility

76Cited by
1References
12Claims
0Family size

Assignee

Inventor

Key dates

Filing dateAug 27, 1992
Grant dateFeb 8, 1994
Priority date
Expiry dateAug 27, 2012

Classification

  • Technology area (CPC A)Human Necessities
  • CPC primaryA61K38/00
  • WIPO fieldPharmaceuticals
  • WIPO sectorChemistry

Abstract

Hydroxy-substituted [(D)Ser].sup.8 -Ciclosporin derivatives, particularly [O-(2-hydroxyethyl)(D)Ser].sup.8 -Ciclosporin, have advantageous pharmacological properties and are useful as immunosuppressants, for example in the treatment of transplant rejection and autoimmune diseases.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.