Patent · US Expired

Chemical process for making angiotesin II antagonist compounds

US5294716A · kind A · utility

7Cited by
0References
9Claims
0Family size

Assignee

Inventors

Key dates

Filing dateJan 17, 1992
Grant dateMar 15, 1994
Priority date
Expiry dateJan 17, 2012

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07D403/10
  • WIPO fieldOrganic fine chemistry
  • WIPO sectorChemistry

Abstract

The invention provides a novel chemical process for the manufacture of quinoline, pyridine and imidazole derivatives of the formula IV wherein Q, Y.sup.1 and Y.sup.2 have the various meanings defined herein, and their non-toxic salts, which are angiotensin II inhibitors. The process involves the removal of an electron-deficient phenyl group or a pyridyl or pyrimidyl group from a compound of the formula VI as defined herein.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.