Patent · US Expired

Stabilization of aminosteroids for topical ophthalmic and other applications

US5332582A · kind A · utility

31Cited by
40References
36Claims
0Family size

Assignee

Inventors

Key dates

Filing dateDec 2, 1992
Grant dateJul 26, 1994
Priority date
Expiry dateDec 2, 2012

Classification

  • Technology area (CPC B)Performing Operations; Transporting
  • CPC primaryB82Y5/00
  • WIPO fieldPharmaceuticals
  • WIPO sectorChemistry

Abstract

The invention provides methods for stabilizing amino-substituted steroid therapeutic agents in topical ophthalmic and other pharmaceutical formulations using effective stabilizing amounts of lightly cross-linked carboxy-containing polymers; Stabilized and stabilized/solubilized pharmaceutical compositions adapted for various routes of administration are also described.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.