Patent · US Expired

Aminoketone derivatives of 1,2-oxazole and use thereof

US5338857A · kind A · utility

7Cited by
0References
7Claims
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Assignee

Inventors

Key dates

Filing dateFeb 24, 1992
Grant dateAug 16, 1994
Priority date
Expiry dateFeb 24, 2012

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07D417/06
  • WIPO fieldOrganic fine chemistry
  • WIPO sectorChemistry

Abstract

Aminoketone derivative compounds containing a heterocyclic ring bonded to an aminoketone moiety and useful as effective ingredients of centrally acting muscle relaxants and pollakiurea curing agents. (+)3-phenyl-5-[2-(1-pyrrolidinylmethyl)butyryl]isoxazole, which has a more remarkable central muscle relaxant action as compared with its racemic modification, can be effectively separated from the racemic modification using optically active 10-camphorsulfonic acid as the agent for the optical resolution.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.