Patent · US Expired

Cycloaminoalkoxyphenyl derivatives, a process for their preparation as well as the compositions containing them

US5340820A · kind A · utility

0Cited by
11References
13Claims
0Family size

Assignee

Inventors

Key dates

Filing dateMar 2, 1992
Grant dateAug 23, 1994
Priority date
Expiry dateMar 2, 2012

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07D471/04
  • WIPO fieldOrganic fine chemistry
  • WIPO sectorChemistry

Abstract

Cycloaminoalkoxyphenyl derivatives useful for the treatment of certain pathological syndromes of the cardiovascular system and ocular diseases of formula: in which: PA0 B represents a --S--, --SO-- or --SO.sub.2 -- group, PA0 R.sub.1 and R.sub.2, which are identical or different, each denotes hydrogen, a methyl or ethyl radical or a halogen such as chlorine, bromine or iodine, PA0 A denotes a straight or linear alkylene radical, having from 2 to 5 carbon atoms or a 2-hydroxypropylene radical in which the hydroxy is optionally substituted by a lower alkyl radical, PA0 Am denotes a group: ##STR1## in which: R.sub.3, R'.sub.3 and R".sub.3, which are identical or different, each denotes hydrogen, a halogen atom such as chlorine or bromine, a lower alkyl group or a lower alkoxy group, R.sub.4 denotes hydrogen or an alkyl radical, PA0 n and m, identical or different, each denotes 0, 1, 2 or 3, PA0 Cy represents a group of formula: ##STR2## pharmaceutically acceptable salts thereof.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.