Patent · US Expired

Imidazolidyl macrolides having immunosuppressive activity

US5344925A · kind A · utility

9Cited by
10References
7Claims
0Family size

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Inventors

Key dates

Filing dateSep 20, 1993
Grant dateSep 6, 1994
Priority date
Expiry dateSep 20, 2013

Classification

  • Technology area (CPC A)Human Necessities
  • CPC primaryA61P37/06
  • WIPO fieldOrganic fine chemistry
  • WIPO sectorChemistry

Abstract

Imidazolidyl macrolides of the general structural Formula I: ##STR1## have been prepared from suitable precursors by alkylation and/or arylation at C-3" and/or C-4" of the cyclohexyl ring. These macrolide immunosuppressants are useful in a mammalian host for the treatment of autoimmune diseases, infectious diseases the prevention of rejection of foreign organ transplants and/or related afflictions, diseases and illnesses.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.