Patent · US Expired

N-(pyrrolo(2,3-d)pyrimidin-3-ylacyl)-glutamic acid derivatives

US5344932A · kind A · utility

55Cited by
3References
7Claims
0Family size

Assignee

Inventor

Key dates

Filing dateMar 22, 1991
Grant dateSep 6, 1994
Priority date
Expiry dateMar 22, 2011

Classification

  • Technology area (CPC Y)Emerging Cross-Sectional Technologies
  • CPC primaryY02P20/582
  • WIPO fieldPharmaceuticals
  • WIPO sectorChemistry

Abstract

N-(Acyl)glutamic acid derivatives in which the acyl group is substituted with 4-hydroxypyrrolo[2,3-d]-pyrimidin-3-yl group are antineoplastic agents. A typical embodiment is N-[4-(2-{4-hydroxy-6-aminopyrrolo-[2,3-d]pyrimidin-3-yl}ethyl)benzoyl]-L-g lutamic acid.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.