Patent · US Expired

Cholesterol-lowering agents

US5369125A · kind A · utility

18Cited by
7References
15Claims
0Family size

Assignee

Inventors

Key dates

Filing dateMar 19, 1993
Grant dateNov 29, 1994
Priority date
Expiry dateMar 19, 2013

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07D493/08
  • WIPO fieldOrganic fine chemistry
  • WIPO sectorChemistry

Abstract

This invention relates to compounds of structural formula (I): ##STR1## which are squalene synthase inhibitors and thus useful as cholesterol lowering agents and antifungal agents. These compounds are also inhibitors of farnesyl protein transferase and farnesylation of the oncogene protein Ras and thus useful in treating cancer.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.