Patent · US Expired

Method of treatment of androgen-related diseases

US5372996A · kind A · utility

48Cited by
17References
29Claims
0Family size

Assignee

Inventor

Key dates

Filing dateOct 19, 1992
Grant dateDec 13, 1994
Priority date
Expiry dateOct 19, 2012

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07J71/001
  • WIPO fieldPharmaceuticals
  • WIPO sectorChemistry

Abstract

A method of treatment of androgen-related diseases such as prostate cancer in susceptible male animals, including humans, comprises administering novel antiandrogens and/or novel sex steroid biosynthesis inhibitors as part of a combination therapy. Sex steroid biosynthesis inhibitors, especially those capable of inhibiting conversion of dehydroepiandrosterone (DHEA) or 4-androstenedione (.DELTA..sup.4 -dione) to natural sex steroida (and testosterone into dihydrotestosterone) in peripheral tissues, are used in combination with antiandrogens usually after blockade of testicular hormonal secretions. Antiestrogens can also be part of the combination therapy. Pharmaceutical compositions and two, three, four and five component kits are useful for such combination treatment.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.