Patent · US Expired

Heterocyclic esters of rapamycin

US5385909A · kind A · utility

166Cited by
27References
15Claims
0Family size

Assignee

Inventors

Key dates

Filing dateNov 22, 1993
Grant dateJan 31, 1995
Priority date
Expiry dateNov 22, 2013

Classification

  • Technology area (CPC A)Human Necessities
  • CPC primaryA61P37/06
  • WIPO fieldPharmaceuticals
  • WIPO sectorChemistry

Abstract

A compound of the structure ##STR1## wherein R and R.sup.1 are each, independently, ##STR2## or hydrogen, R.sup.2 is a heterocyclic radical which may be optionally substituted; PA1 n=0-6; with the proviso that R and R.sup.1 are both not hydrogen, or a pharmaceutically acceptable salt thereof which is useful as an immunosuppressive, antiinflammatory, antifungal, antiproliferative, and antitumor agent.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.