Patent · US Expired

2-saccharinylmethyl aryl and aryloxy acetates useful as proteolytic enzyme inhibitors

US5385923A · kind A · utility

2Cited by
12References
13Claims
0Family size

Assignee

Inventors

Key dates

Filing dateAug 20, 1993
Grant dateJan 31, 1995
Priority date
Expiry dateAug 20, 2013

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07D513/04
  • WIPO fieldPharmaceuticals
  • WIPO sectorChemistry

Abstract

4-R.sup.4 --R.sup.5 -2-Saccharinylmethyl aryl and aryloxy acetates, useful in the treatment of degenerative diseases, are prepared by reacting a 4-R.sup.4 --R.sup.5 -2-halomethylsaccharin with an aryl or aryloxyacetic acid in the presence of an acid-acceptor.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.