Patent · US Expired

Monospecific antibodies and assay system for detecting stromelysin cleavage products

US5387504A · kind A · utility

12Cited by
1References
9Claims
0Family size

Assignee

Inventors

Key dates

Filing dateSep 30, 1992
Grant dateFeb 7, 1995
Priority date
Expiry dateSep 30, 2012

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07K16/18
  • WIPO fieldBiotechnology
  • WIPO sectorChemistry

Abstract

Monospecific antibodies are produced which are specific for fragments of the connective tissue protein aggrecan, generated by specific stromelysin cleavage. These monospecific antibodies are used in an assay system to detect polypeptide fragments of aggrecan, produced by the specific cleavage of aggrecan by stromelysin. The presence of aggrecan polypeptide fragments demonstrates stromelysin activity. Elevations of stromelysin occur in osteoarthritis, rheumatoid arthritis, atherosclerotic lesions, gout, inflammatory bowel disease (IBD), idiopathic pulmonary fibrosis (IPF), certain cancers, joint injuries, and numerous inflammatory diseases. The monospecific antibodies and the assay system are used to quantitate aggrecan polypeptide fragments as a readout of stromelysin activity and to evaluate potential stromelysin inhibitors.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.