Aminobenzoic acid derivatives useful for treating gastro-intestinal conditions
US5389643A · kind A · utility
Assignee
Inventors
Key dates
| Filing date | Feb 3, 1993 |
| Grant date | Feb 14, 1995 |
| Priority date | — |
| Expiry date | Feb 3, 2013 |
Classification
- Technology area (CPC A)Human Necessities
- CPC primaryA61P43/00
- WIPO fieldPharmaceuticals
- WIPO sectorChemistry
Abstract
An aminobenzoic acid derivative represented by the following general formulas (I), (I-2) or (I-3), or a pharmacologically acceptable salt thereof, which exhibits a serotonin antagonism and an acetylcholine release accelerating activity at a well-balanced activity ratio and which is efficacious as a drug for patients with gastrointestinal unindentified complaints: ##STR1## wherein R.sup.1 represents a group such as an alkynyl or cyanoalkyl group; R.sup.2 represents a group such as an amino or acylamino group; PA1 R.sup.3 represents a halogen atom; PA1 X represents --O-- or --NH--; and PA1 A represents an oxygen or sulfur atom.
Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.