Patent · US Expired

Fused benzeneoxyacetic acid derivatives

US5389666A · kind A · utility

5Cited by
5References
12Claims
0Family size

Assignee

Inventors

Key dates

Filing dateDec 28, 1992
Grant dateFeb 14, 1995
Priority date
Expiry dateDec 28, 2012

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07D401/06
  • WIPO fieldOrganic fine chemistry
  • WIPO sectorChemistry

Abstract

A fused benzeneoxyacetic acid derivative of the formula (I): ##STR1## R.sup.1 is OH, alkoxy, (alkyl)amino, residue of an amino acid; A is phenyl, alkyl substituted by phenyl, residue of an imidazole, imidazole-2-yloxy(thio), 2-oxoimidazole, pyrazole, oxadiazole, oxazole, triazole, isoxazole or isothiazole, in the group of benzene may be substituted by one to three of alkyl, alkoxy, halogen, nitro or trihalomethyl; PA1 e is 3-5; PA1 f is 1-3; PA1 p is 1-4; PA1 q is 0-2; PA1 r is 1-4; PA1 s is 0-3) and salts thereof possess an agonistic on PGI.sub.2 receptor, so it is useful for prevention and/or treatment of thrombosis, arteriosclerosis, inchemic heart diseases, gastric alcer and hypertention.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.