Patent · US Expired

Quinoline derivatives and processes for preparing the same

US5409933A · kind A · utility

7Cited by
10References
5Claims
0Family size

Inventors

Key dates

Filing dateJun 8, 1993
Grant dateApr 25, 1995
Priority date
Expiry dateJun 8, 2013

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07D487/04
  • WIPO fieldOrganic fine chemistry
  • WIPO sectorChemistry

Abstract

The present invention relates to novel quinoline derivatives of formula (I): ##STR1## wherein R.sub.1, R.sub.2, R.sub.3, X, Y and Z are defined as in the specification, and pharmaceutically acceptable acid addition salts thereof, and also to processes for preparing these compounds. The present invention also provides an antibacterial composition comprising a compound of formula (I) or its acid addition salt as an active ingredient and pharmaceutically acceptable excipient. The novel quinoline derivatives of the present invention have an excellent antibacterial activity against bacteria or bacteroides.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.