Patent · US Expired

Isoxazole, isothiazole and pyrazole compounds that enhance cognitive function

US5409946A · kind A · utility

28Cited by
0References
13Claims
0Family size

Assignee

Inventors

Key dates

Filing dateSep 8, 1993
Grant dateApr 25, 1995
Priority date
Expiry dateSep 8, 2013

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07D413/04
  • WIPO fieldPharmaceuticals
  • WIPO sectorChemistry

Abstract

Novel isoxazole isothiazole and pyrazole compounds of the formula: ##STR1## wherein A, R.sup.1, and R.sup.2 are specifically defined, or pharmaceutical salts thereof, are selective and potent cholinergic ligands at neuronal nicotinic receptors, useful in the treatment of cognitive, neurological and mental disorders characterized by decreased cholinergic function, as well as in the treatment of alcohol intoxication and petit real absence epilepsy.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.