Patent · US Expired

2-thienylimidazo[2,1-.beta.]benzothiazole-3-acetic acid derivatives, their preparation and their use

US5418248A · kind A · utility

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1References
4Claims
0Family size

Assignee

Inventors

Key dates

Filing dateDec 29, 1993
Grant dateMay 23, 1995
Priority date
Expiry dateDec 29, 2013

Classification

  • Technology area (CPC A)Human Necessities
  • CPC primaryA61P25/20
  • WIPO fieldPharmaceuticals
  • WIPO sectorChemistry

Abstract

Compounds of the formula: ##STR1## in which R.sub.1 represents a hydroxy group, a C.sub.1 -C.sub.4 alkoxy group or an amino group of general formula --NR.sub.4 R.sub.5 in which R.sub.4 and R.sub.5 each represent, independently of each other, a hydrogen atom, a straight or branched C.sub.1 -C.sub.4 alkyl group, an allyl group or a methoxyethyl group, or alternatively --NR.sub.4 R.sub.5 represents a heterocycle containing 3 to 6 carbon atoms, PA0 Y represents a thienyl group optionally substituted by an alkyl group, and PA0 X represents a hydrogen or halogen atom, are useful as anticonvulsants and auxiolytics.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.