Patent · US Expired

9-deoxotaxane compounds

US5440056A · kind A · utility

52Cited by
1References
10Claims
0Family size

Assignee

Inventors

Key dates

Filing dateMar 9, 1994
Grant dateAug 8, 1995
Priority date
Expiry dateMar 9, 2014

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07D305/14
  • WIPO fieldOrganic fine chemistry
  • WIPO sectorChemistry

Abstract

Compounds having the formula ##STR1## wherein --OR.sup.1 comprises alkanoyl or the C-13 side-chain of taxol; R.sup.2, R.sup.3, and R.sup.6 can be oxygenated or hydrogen in various combinations; and R.sup.4 and R.sup.5 are acyl groups, as well as a process for the preparation thereof, pharmaceutical compositions containing the above compounds, and a method for their use in inhibiting tumor growth.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.