Patent · US Expired

Method of treatment of neurodegeneration with calpain inhibitors

US5444042A · kind A · utility

31Cited by
39References
35Claims
0Family size

Assignees

Inventors

Key dates

Filing dateMar 7, 1994
Grant dateAug 22, 1995
Priority date
Expiry dateMar 7, 2014

Classification

  • Technology area (CPC A)Human Necessities
  • CPC primaryA61K31/535
  • WIPO fieldPharmaceuticals
  • WIPO sectorChemistry

Abstract

The present invention provides a method of treating a neurodegenerative pathology in a human patient. This method includes selecting a patient for monitoring for the presence of a neurodegenerative pathology associated with enhanced Calpain activity and monitoring the patient for indicia of the onset or existence of such a pathology. In response to the detection of any such indicium of the presence or onset of the pathology, a therapeutically efficacious amount of a Peptide Ketoamide compound, or a pharmaceutically acceptable salt or derivative thereof, together with a pharmaceutically acceptable carrier is administered. The invention also provides additional methods of treatment and pharmaceutical compositions using Peptide Ketoamides, Peptide Ketoacids and Peptide Ketoesters.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.