Patent · US Expired

Benzothiophene compounds, intermediates, compositions, and methods

US5510498A · kind A · utility

18Cited by
13References
23Claims
0Family size

Assignee

Inventor

Key dates

Filing dateJun 6, 1995
Grant dateApr 23, 1996
Priority date
Expiry dateJun 6, 2015

Classification

  • Technology area (CPC Y)Emerging Cross-Sectional Technologies
  • CPC primaryY02P20/55
  • WIPO fieldPharmaceuticals
  • WIPO sectorChemistry

Abstract

The present invention provides compounds of formula II ##STR1## wherein R.sup.1a is --H or --OR.sup.7 in which R.sup.7 is a hydroxy protecting group; PA1 R.sup.2a is --H, halo, or --OR.sup.8 in which R.sup.8 is a hydroxy protecting group, providing when Z is --S--, R.sup.2a is not halo; PA1 R.sup.6 is --H or a hydroxy protecting group which can be selectively removed; and PA1 Z is --O-- or --S--; or a pharmaceutically acceptable salt thereof, which are useful intermediates for the preparation of biologically active compounds.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.