Patent · US Expired

Peptidyl ketoamides

US5514694A · kind A · utility

46Cited by
1References
14Claims
0Family size

Assignee

Inventors

Key dates

Filing dateJun 24, 1993
Grant dateMay 7, 1996
Priority date
Expiry dateJun 24, 2013

Classification

  • Technology area (CPC A)Human Necessities
  • CPC primaryA61K38/00
  • WIPO fieldPharmaceuticals
  • WIPO sectorChemistry

Abstract

A novel class of peptide .alpha.-ketoamides useful for selectively inhibiting serine proteases, selectively inhibiting cysteine proteases, generally inhibiting all serine proteases, and generally inhibiting all cysteine proteases, having the formula Y--CO--AA.sup.2 --AA.sup.1 --CO--NH--X. Processes for the synthesis of peptidyl .alpha.-ketoamide derivatives.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.