Patent · US Expired

Substituted imidazolyl-alkyl-piperazine and -diazepine derivatives

US5514800A · kind A · utility

0Cited by
5References
10Claims
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Assignee

Inventors

Key dates

Filing dateSep 20, 1993
Grant dateMay 7, 1996
Priority date
Expiry dateSep 20, 2013

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07D403/06
  • WIPO fieldOrganic fine chemistry
  • WIPO sectorChemistry

Abstract

Substituted imidazolyl-alkyl-piperazine and diazepine derivatives of Formula A: ##STR1## wherein R.sup.1, R.sup.2, R.sup.3, R.sup.4, R.sup.5, m, n and q are defined as in the specification, and the pharmaceutically acceptable salts thereof. The compounds have calcium entry blocking activity with selectivity for cerebral blood vessels, and have protective activity against some of the deleterious effects resultant upon cerebral ischemia.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.