Patent · US Expired

Certain tetrahydrocannabinol-7-oic acid derivatives

US5538993A · kind A · utility

74Cited by
5References
24Claims
0Family size

Assignee

Inventors

Key dates

Filing dateFeb 7, 1994
Grant dateJul 23, 1996
Priority date
Expiry dateFeb 7, 2014

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07D311/80
  • WIPO fieldOrganic fine chemistry
  • WIPO sectorChemistry

Abstract

The invention relates to compounds of the formula ##STR1## having the (3S,4S) configuration and being essentially free of the (3R,4R) enantiomer, in which A--B indicates an optional 1(2) or 6(1) double bond, X is carboxy, carbalkoxy, or carboxamido, linked to the ring directly or through an alkylene linkage, G is halogen, alkyl, or oxy, and Y is alkyl, oxy, or oxyalkylene. The invention further relates to the synthesis of such compounds, and to pharmaceutical compositions and therapeutic methods in which such compounds may be employed.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.