Patent · US Expired

Melatonergic agents

US5541228A · kind A · utility

16Cited by
14References
17Claims
0Family size

Assignee

Inventors

Key dates

Filing dateMar 8, 1995
Grant dateJul 30, 1996
Priority date
Expiry dateMar 8, 2015

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07C2601/08
  • WIPO fieldPharmaceuticals
  • WIPO sectorChemistry

Abstract

New melatonergic agents are phenyl alkanyl or phenyl alkyl substituted carboxamides and ureas of Formula I: ##STR1## wherein: R.sub.1 =C.sub.1-3 alkyl, allyl, C.sub.3-6 cycloalkyl substituted C.sub.1-4 alkyl; PA1 R.sub.2 =hydrogen, halogen or C.sub.1-4 alkoxy; PA1 R.sub.3 =hydrogen or C.sub.1-4 alkyl; PA1 R.sub.4 =C.sub.1-4 alkyl, C.sub.1-4 alkyl substituted amino, carboxylic acid substituted PA1 C.sub.1-4 alkyl or C.sub.3-6 cycloalkyl, C.sub.3-6 cycloalkyl, or straight or branched chain C.sub.2-4 alkenyl; PA1 A=a linear C.sub.2-4 alkanediyl or alkenediyl chain, provided that A not be --CH.sub.2 CH.sub.2 -- when X is a bond; and PA1 X=a covalent bond or oxygen.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.