Patent · US Expired

Bisarylcarbinol derivatives as inhibitors of leukotriene biosynthesis

US5552437A · kind A · utility

7Cited by
0References
9Claims
0Family size

Assignee

Inventors

Key dates

Filing dateOct 27, 1994
Grant dateSep 3, 1996
Priority date
Expiry dateOct 27, 2014

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07D417/14
  • WIPO fieldOrganic fine chemistry
  • WIPO sectorChemistry

Abstract

Compounds having the Formula I: EQU R.sup.1 R.sup.2 C(OR.sup.3)--Ar.sup.1 --X--Ar.sup.2 --Ar.sup.3I re inhibitors of leukotriene biosynthesis. These compounds are useful as anti-asthmatic, anti-allergic, anti-inflammatory, and cytoprotective agents. They are also useful in treating angina, cerebral spasm, glomerular nephritis, hepatitis, endotoxemia, uveitis, and allograft rejection and in preventing the formation of atherosclerotic plaques.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.