Carboxamide derivatives for treating asthma
US5559132A · kind A · utility
11Cited by
9References
11Claims
0Family size
Assignee
Inventor
Key dates
| Filing date | Feb 21, 1995 |
| Grant date | Sep 24, 1996 |
| Priority date | — |
| Expiry date | Feb 21, 2015 |
Classification
- Technology area (CPC C)Chemistry; Metallurgy
- CPC primaryC07D211/86
- WIPO fieldOrganic fine chemistry
- WIPO sectorChemistry
Abstract
The present invention concerns novel carboxamide derivatives of formula I, set out hereinbelow which antagonize the pharmacological actions of one of the endogenous neuropeptide tachykinins at the neurokinin 2 (NK2) receptor, making them useful whenever such antagonism is desired, such as in the treatment of asthma and related conditions. The invention also provides pharmaceutical compositions containing the novel carboxamide derivatives for use in such treatment, methods for their use, and processes and intermediates for the manufacture of the novel carboxamide derivatives. ##STR1##
Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.