Patent · US Expired

Polypeptide capable of interacting with thrombin

US5574007A · kind A · utility

14Cited by
0References
12Claims
0Family size

Assignee

Inventors

Key dates

Filing dateJun 15, 1994
Grant dateNov 12, 1996
Priority date
Expiry dateJun 15, 2014

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC12N15/80
  • WIPO fieldBiotechnology
  • WIPO sectorChemistry

Abstract

Disclosed is a substantially pure polypeptide having a specific amino acid sequence containing (a) an amino acid residue selected from the group consisting of Asp, Glu and Gla wherein Gla represents a .gamma.-carboxyglutamic acid residue or (b) a peptide or polypeptide residue consisting of at least two amino acid residues selected from Asp, Glu and Gla, wherein the above-mentioned at least two amino acid residues are all the same or combinations of the Asp, Glu and Gla. The polypeptide is capable of interacting with thrombin to form a binding therebetween, thereby exhibiting an activity to inhibit the blood coagulation and platelet aggregation by thrombin and/or an activity to promote the thrombin-catalyzed activation of protein C. This novel polypeptide has a low molecular weight so that it is suitable for oral or nasal administration.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.