Patent · US Expired

Process for the preparation of Baccatin III and 10-deacetylbaccatin III derivatives

US5578739A · kind A · utility

9Cited by
1References
10Claims
0Family size

Assignee

Inventor

Key dates

Filing dateJul 6, 1995
Grant dateNov 26, 1996
Priority date
Expiry dateJul 6, 2015

Classification

  • Technology area (CPC Y)Emerging Cross-Sectional Technologies
  • CPC primaryY02P20/55
  • WIPO fieldOrganic fine chemistry
  • WIPO sectorChemistry

Abstract

This invention relates to process for the preparation of a taxane derivative of general formula (I): ##STR1## and use of the product obtained for the preparation of taxane derivatives of general formula (II): ##STR2## In the general formula (I), R.sub.1 is an acetyl radical or a protective grouping G.sub.1 is a protective grouping and R is a t-butoxy or phenyl radical. In the general formula (II), R is a t-butoxy or phenyl radical and R'.sub.1 is a hydrogen atom or an acetyl radical.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.