Patent · US Expired

Prodrugs for antibody directed enzyme prodrug therapy

US5587161A · kind A · utility

26Cited by
1References
21Claims
0Family size

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Inventors

Key dates

Filing dateDec 21, 1994
Grant dateDec 24, 1996
Priority date
Expiry dateDec 21, 2014

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07C311/51
  • WIPO fieldPharmaceuticals
  • WIPO sectorChemistry

Abstract

Prodrugs, of generic formula I, are disclosed for use in antibody directed enzyme prodrug therapy (ADEPT). The prodrugs substrates for carboxypeptidase G2 (CPG2) and yield more cytotoxic drugs than known products of CPG2 catalysed

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.