Patent · US Expired

Pyridyl-propan-2-yl esters of 1-adamantane carboxylates

US5595995A · kind A · utility

5Cited by
0References
10Claims
0Family size

Assignee

Inventors

Key dates

Filing dateJan 18, 1995
Grant dateJan 21, 1997
Priority date
Expiry dateJan 18, 2015

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07D213/55
  • WIPO fieldPharmaceuticals
  • WIPO sectorChemistry

Abstract

Compounds having the general formula: ##STR1## wherein each of R.sup.1 and R.sup.2 independently represents hydrogen or alkyl of 1 to 4 carbon atoms; A represents --O-- or --CR.sup.4 R.sup.5, where R.sup.4 and R.sup.5 are defined as for R.sup.1 or R.sup.2 ; R.sup.3 represents an adamantyl group; and Py represents a 3- or 4-pyridyl group, as free bases or their pharmaceutically acceptable salts are useful in treating androgen-dependent, especially prostatic, cancer.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.