Selective antagonists for GABA.sub.rho receptor
US5627169A · kind A · utility
3Cited by
0References
9Claims
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Key dates
| Filing date | Jul 20, 1994 |
| Grant date | May 6, 1997 |
| Priority date | — |
| Expiry date | Jul 20, 2014 |
Classification
- Technology area (CPC C)Chemistry; Metallurgy
- CPC primaryC07F9/59
- WIPO fieldOrganic fine chemistry
- WIPO sectorChemistry
Abstract
Novel phosphinic and phosphonic acid derivatives of pyridine, pyrrole and azepine with utility as antagonists of the GABA.sub.rho receptor are disclosed. These compounds have utility as modulators of the excitability of the central nervous system as mediated by their ability to specifically act on closed-channel binding sites of GABA.sub.rho receptors.
Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.