Patent · US Expired

Method of forming amino acid-derived diaminopropanols useful as chemical intermediates for protease-inhibitors

US5631405A · kind A · utility

13Cited by
9References
10Claims
0Family size

Assignee

Inventors

Key dates

Filing dateJun 7, 1995
Grant dateMay 20, 1997
Priority date
Expiry dateJun 7, 2015

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07D207/12
  • WIPO fieldOrganic fine chemistry
  • WIPO sectorChemistry

Abstract

The present invention relates to a method of forming a 1,3-diamino-3-substituted-2-propanol chemical intermediate from which various chemicals, such as selected protease-inhibitors and other drugs, as well as polymers, can be synthesized. This method includes contacting a nitromethyl amino acid compound with at least one reducing agent to form the 1,3-diamino-3-substituted-2-propanol chemical intermediate.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.