Patent · US Expired

(Z,Z), (Z,E) and (E,Z) isomers of substituted bis(phenylmethylene)cycloketones

US5633381A · kind A · utility

24Cited by
2References
23Claims
0Family size

Assignee

Inventors

Key dates

Filing dateJul 5, 1994
Grant dateMay 27, 1997
Priority date
Expiry dateJul 5, 2014

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07D335/02
  • WIPO fieldOrganic fine chemistry
  • WIPO sectorChemistry

Abstract

This invention relates to novel (Z,Z), (Z,E) and (E,Z) olefin isomers of substituted benzylidene cycloketones and their pharmaceutically acceptable salts. The compounds of the invention are potent factor Xa inhibitors thereby acting as anticoagulants useful in a number of thrombotic disease states. Pharmaceutical compositions are proposed for the compounds.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.