Patent · US Expired

Substituted pyrrolidin-3-yl-alkyl-piperidines

US5635510A · kind A · utility

14Cited by
3References
57Claims
0Family size

Assignee

Inventors

Key dates

Filing dateOct 31, 1994
Grant dateJun 3, 1997
Priority date
Expiry dateOct 31, 2014

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07D471/10
  • WIPO fieldOrganic fine chemistry
  • WIPO sectorChemistry

Abstract

The present invention relates to substituted pyrrolidinyl-3-yl-alkyl-piperidines, their stereoisomers, and pharmaceutically acceptable salts thereof and processes for preparation of the same. The compounds of the present invention are useful in their pharmacological activities such as tachykinin antagonism, especially substance P and neurokinin A antagonism, and the like. Compounds having the property of tachykinin antagonism are indicated for conditions associated with neurogenic inflammation and other diseases described herein.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.