Patent · US Expired

Polyamine derivatives as antineoplastic agents

US5654484A · kind A · utility

7Cited by
0References
5Claims
0Family size

Assignee

Inventors

Key dates

Filing dateJun 1, 1995
Grant dateAug 5, 1997
Priority date
Expiry dateJun 1, 2015

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07C211/09
  • WIPO fieldOrganic fine chemistry
  • WIPO sectorChemistry

Abstract

The present invention relates to a method for the treatment of patients suffering from certain neoplastic disease states which comprises administering a therapeutically effective amount of a compound of the formula: ##STR1## wherein m is an integer 6 to 9, Z is a saturated (C.sub.2 -C.sub.6) alkylene moiety, each R group independently is hydrogen, methyl, ethyl, or n-propyl except that both R groups cannot be hydrogen when Z is a straight chain; or a pharmaceutically acceptable acid addition salt thereof. Said treatment can optionally comprise conjunctive therapy with a polyamine oxidase inhibitor. The invention also relates to certain novel polyamine derivatives.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.