Patent · US Expired

Compositions and methods for treating mast-cell mediated conditions

US5656660A · kind A · utility

8Cited by
0References
42Claims
0Family size

Assignee

Inventors

Key dates

Filing dateMay 31, 1995
Grant dateAug 12, 1997
Priority date
Expiry dateMay 31, 2015

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07C2601/14
  • WIPO fieldPharmaceuticals
  • WIPO sectorChemistry

Abstract

The present invention describes compounds, methods and compositions effective to treat mast cell mediated inflammatory conditions, such as conjunctivitis, asthma and allergic rhinitis. The compounds of the invention comprise novel mono- and di-aminomethylbenzyl, aminobenzyl, guanidylbenzyl and benzyl tryptase inhibitors. The compositions for treating mast cell mediated inflammatory conditions include oral, inhalant and topical preparations as well as devices comprising such preparations.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.