Patent · US Expired

Opioid diarylmethylpiperazines and piperdines

US5658908A · kind A · utility

42Cited by
4References
26Claims
0Family size

Assignee

Inventors

Key dates

Filing dateAug 3, 1994
Grant dateAug 19, 1997
Priority date
Expiry dateAug 3, 2014

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07K5/06078
  • WIPO fieldPharmaceuticals
  • WIPO sectorChemistry

Abstract

Diarylmethylpiperazine compounds having utility as receptor-binding species, e.g., for mediating analgesia, and for combatting drug addiction, alcohol addiction, and drug overdose. The compounds may be administered orally, rectally, topically, nasally, ophthalmically, or parenterally (subcutaneously, intramuscularly, and intravenously), for veterinary and human use, and include delta receptor and mu receptor binding species.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.