Patent · US Expired

2-imidazolinylamino heterocyclic compounds useful as alpha-2 adrenoceptor agonists

US5663189A · kind A · utility

8Cited by
3References
22Claims
0Family size

Assignee

Inventors

Key dates

Filing dateJun 7, 1995
Grant dateSep 2, 1997
Priority date
Expiry dateJun 7, 2015

Classification

  • Technology area (CPC A)Human Necessities
  • CPC primaryA61K31/4178
  • WIPO fieldPharmaceuticals
  • WIPO sectorChemistry

Abstract

The subject invention relates to compounds having the structure: ##STR1## wherein (a) n is an integer from 1 to about 3; PA1 (b) X and Y are each independently selected from O, S and CH.sub.2, with at least one of X and Y being O or S; PA1 (c) R is unsubstituted, straight or branched chain alkanyl or alkanoxy having from 1 to about 3 non-hydrogen atoms; and PA1 (d) R' is selected from hydrogen, methyl, cyano, and halo; pharmaceutical compositions containing such compounds; and the use of such compounds for preventing or treating one or more of respiratory disorders, ocular disorders, and gastrointestinal disorders.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.