Patent · US Expired

Substituted 1,4-diazapine caprolactams useful for treatment of HIV disease

US5663333A · kind A · utility

5Cited by
3References
15Claims
0Family size

Assignee

Inventors

Key dates

Filing dateMar 30, 1993
Grant dateSep 2, 1997
Priority date
Expiry dateMar 30, 2013

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07D281/06
  • WIPO fieldOrganic fine chemistry
  • WIPO sectorChemistry

Abstract

This invention relates to novel substituted caprolactams, including 4-azacaprolactams, and derivatives thereof which inhibit HIV protease and are useful for treatment of HIV disease. Also included in this invention are pharmaceutical compositions containing such caprolactams, and to methods of using such caprolactams for the treatment of HIV disease.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.