Patent · US Expired

Anti-cancer composition comprising rhodacyanine compound and cyclodextrin

US5670530A · kind A · utility

10Cited by
1References
19Claims
0Family size

Assignees

Inventors

Key dates

Filing dateJun 7, 1995
Grant dateSep 23, 1997
Priority date
Expiry dateJun 7, 2015

Classification

  • Technology area (CPC B)Performing Operations; Transporting
  • CPC primaryB82Y5/00
  • WIPO fieldPharmaceuticals
  • WIPO sectorChemistry

Abstract

An anti-cancer composition comprising a rhodacyanine compound and cyclodextrin or derivative thereof, wherein said rhodacyanine compound is selected from the group consisting of compounds represented by the following Formula (I), the cation moiety of which has a log P value of 4.5-12: ##STR1## wherein X.sub.1 and X.sub.2, which may be the same or different, each represents O, S, Se, ##STR2## Y.sub.1 represents O, S, Se, or ##STR3## R.sub.1 and R.sub.3, which may be the same or different, each represents an alkyl group; R.sub.2 represents an alkyl group, an aryl group or a heterocyclic group; Z.sub.1 and Z.sub.2, which may be the same or different, each represents an atomic group necessary to form a 5- or 6-membered ring; L.sub.1, L.sub.2 and L.sub.3, which may be the same or different, each represents a methine group or nitrogen atom and L.sub.1 and R.sub.3 may combine and form a 5- or 6-membered ring; R.sub.4 and R.sub.5, which may be the same or different, each represents an alkyl group; R.sub.6 and R.sub.7, which may be the same or different, each represents an alkyl group or an aryl group; Q represents a pharmaceutically acceptable anion; j and k, which may be the same or diffe…

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.