Patent · US Expired

Process for preparing 7-trialkylsilyl baccatin III

US5670658A · kind A · utility

10Cited by
4References
10Claims
0Family size

Assignee

Inventors

Key dates

Filing dateOct 3, 1996
Grant dateSep 23, 1997
Priority date
Expiry dateOct 3, 2016

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07F7/188
  • WIPO fieldOrganic fine chemistry
  • WIPO sectorChemistry

Abstract

The present invention relates to a novel process for the preparation of 7-trialkylsilylbaccatin III of general formula: ##STR1## in which the symbols R, which may be identical or different, represent alkyl radicals containing 1 to 4 carbon atoms which are optionally substituted with a phenyl radical, starting with 10-deacetylbaccatin III of formula: ##STR2## In the general formula (I), each of the symbols R preferably represents a straight or branched alkyl radical containing 1 to 4 carbon atoms. Even more particularly, each of the symbols R represents an ethyl radical.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.