Patent · US Expired

Antihypercholesterolemic compounds and related pharmaceutical compositions and methods of use

US5688780A · kind A · utility

2Cited by
4References
17Claims
0Family size

Assignee

Inventors

Key dates

Filing dateFeb 29, 1996
Grant dateNov 18, 1997
Priority date
Expiry dateFeb 29, 2016

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07J71/0042
  • WIPO fieldOrganic fine chemistry
  • WIPO sectorChemistry

Abstract

Novel antihypercholesterolemic agents are provided. An exemplary group of compounds has the structural formula (I) ##STR1## wherein R is a C-17 side chain, R.sup.1 is --OH, .dbd.O, or the like, and X and Y are CH, C--OH, C--OCH.sub.3 or C--Z. Methods of using the compound of formula (I) or other novel oxysterol analogs to treat hypercholesterolemia are provided, as are pharmaceutical compositions containing the compounds.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.