Patent · US Expired

Process for the preparation of substituted thiopyran-1-oxides

US5688954A · kind A · utility

0Cited by
1References
11Claims
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Assignee

Inventors

Key dates

Filing dateApr 24, 1996
Grant dateNov 18, 1997
Priority date
Expiry dateApr 24, 2016

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07D213/32
  • WIPO fieldOrganic fine chemistry
  • WIPO sectorChemistry

Abstract

A process is described for the preparation of a compound of formula (IX) from 4-hydroxybutyl 3-pyridyl ketone. The compound of formula (IX) is an intermediate useful in the preparation of (1R,2R)-2-(3-pyridyl)-N-alkyl-tetrahydro-2H-thiopyran-2-carbothioamide 1-oxides which possess useful pharmaceutical properties, for example anti-hypertensive properties. ##STR1##

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.