Patent · US Expired

Pseudopeptides derived from neurokinins

US5708016A · kind A · utility

1Cited by
0References
9Claims
0Family size

Assignee

Inventors

Key dates

Filing dateFeb 14, 1997
Grant dateJan 13, 1998
Priority date
Expiry dateFeb 14, 2017

Classification

  • Technology area (CPC A)Human Necessities
  • CPC primaryA61K38/00
  • WIPO fieldPharmaceuticals
  • WIPO sectorChemistry

Abstract

A compound of formula (I): ##STR1## in which: R.sub.1 represents an indolyl, naphthyl, tetrahydronaphthyl, thienyl, phenyl, optionally substituted, or (C.sub.3 -C.sub.7)cycloalkyl group, PA1 n represents an integer such that 1.ltoreq.n.ltoreq.8, PA1 m represents an integer such that 1.ltoreq.m.ltoreq.4, PA1 R.sub.2 represents an unsubstituted or substituted benzyl group, an unsubstituted or substituted phenyl group or a linear or branched (C.sub.1 -C.sub.6)alkyl group, its enantiomers, diastereoisomers and epimers as well as its addition salts with a pharmaceutically acceptable acid or base, and medicinal products containing the same are useful as substance P antagonists.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.